| Original document(43 pages) 中文版 |
Pyrimidine derivatives of general formula (I) or nontoxic salts thereof, useful as intermediates for the synthesis of drugs and/or as drugs, particularly elastase inhibitors. In formulas (I), R<1> is H or F; R<2> is -CH(OR<3>)2, CHO, COOH, alkoxycarbonyl, furan-2-yl, a group of general formula (II), or the like; R<3> is Me or Et; and R<4> is alkyl, phenyl, (substituted) benzyl, or the like. |
Application Number
申请号 |
00816305 |
Application Date
申请日 |
2000.09.26 |
| Title 名称 |
Pyrimidine derivatives, process for preparing the derivatives and drugs containing the same as active ingredient |
Publication Number
公开号 |
1399632 |
Publication Date
公开日 |
2003.02.26 |
| Approval Pub. Date |
|
Granted Pub. Date |
|
| International Classification 分类号 |
A61K31/505;A61K31/506;A61P1/02;A61P9/00;A61P11/00;C07D239/36;C07D405/06;C07D413/12 |
Applicant(s) Name
申请人 |
Ono Pharmaceutical Co., Ltd. |
| Address 地址 |
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| Inventor(s) Name 发明人 |
Kojima Tsutomu;Okada Takanori;Hachiya Katsutoshi |
| Attorney & Agent 代理人 |
cao wen yang liqin |
| More information 更 多 信 息 |
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