The present invention provides one kind of polyene taxol liposome capable of being used for injection and oral taking and its solid preparation, and features that polyene taxol is coated with phospholipid matter and additive so as to prepare polyene taxol liposome preparation with small size, high coating rate, high stability and less toxic side effect. The polyene taxol liposome of the present invention has raised targeting effect on cancer cell, enhanced tumor cell killing effect, high curative effect and less toxic side effect. The present invention also provides several preparation processes of polyene taxol liposome, and the preparation processes are simple, low in cost and suitable for industrial production. |