Original document(13 pages)  中文版
    This invention provides a salt that is produced by [(R)-[(1S)-2-methyl-1- (1-keto-propoxy)propoxy](4-benzene butyl) oxygen phosphino]acetic acid and 10,11-di-H Cinchonidine, its structure is shown by formula(1). This invention also provides preparation of using this salt to optically split racemoid which consists of [(R)-[(1S)-2-methyl-1-(1-keto-propoxy)propoxy](4-benzene butyl) oxygen phosphino] acetic acid and [(S)-[(1R)-2-methyl-1-(1-keto-propoxy) propoxy](4- benzene butyl) oxygen phosphino] acetic acid. Compared with present resolution preparation, the yield and optical purity of resolution is obviously raised, it needs not recryst many times to depurate, and dosis of resolution agent is reduced.
Application Number
申请号
200510030872 Application Date
申请日
2005.10.27
Title 名称 Optical active substitution oxyphosphonate salt acetate and its use
Publication Number
公开号
1955185 Publication Date
公开日
2007.05.02
Approval Pub. Date Granted Pub. Date
International Classification 分类号 C07F9/32;C07D401/14
Applicant(s) Name
申请人
Shanghai Medical Industry Inst.
Address 地址
Inventor(s) Name 发明人 Zhang Qingwen;Diao Yuanyuan;Xu Yanyan;Shi Huilin
Attorney & Agent 代理人 louxian yang
More information 更  多  信  息


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